Antineoplastic Agents, Hormonal

Name
Antineoplastic Agents, Hormonal
Accession Number
DBCAT000063
Description

Antineoplastic agents that are used to treat hormone-sensitive tumors. Hormone-sensitive tumors may be hormone-dependent, hormone-responsive, or both. A hormone-dependent tumor regresses on removal of the hormonal stimulus, by surgery or pharmacological block. Hormone-responsive tumors may regress when pharmacologic amounts of hormones are administered regardless of whether previous signs of hormone sensitivity were observed. The major hormone-responsive cancers include carcinomas of the breast, prostate, and endometrium; lymphomas; and certain leukemias. (From AMA Drug Evaluations Annual 1994, p2079)

Drugs
Drug Drug Description
Leuprolide A peptide-based GnRH receptor superagonist used for the palliative treatment of prostate cancer, uterine leiomyomata, endometriosis, and central precocious puberty.
Goserelin A synthetic analog of luteinizing hormone-releasing hormone used to treat breast cancer and prostate cancer by reducing secretion of gonadotropins from the pituitary.
Octreotide A peptide drug used to treat acromegaly as well as diarrhea associated with metastatic carcinoid tumors and vasoactive intestinal peptide secreting tumors.
Diethylstilbestrol Used in the treatment of prostate cancer. Previously used in the prevention of miscarriage or premature delivery in pregnant women prone to miscarriage or premature delivery.
Chlorotrianisene Used to treat symptoms of menopause, deficiencies in ovary function (including underdevelopment of female sexual characteristics and some types of infertility), and in rare cases, prostate cancer. Chlorotrianisene may also...
Megestrol acetate A progestin that is administered orally to treat anorexia and cachexia or serious unexplained weight loss and is also used as an antineoplastic agent to treat certain types of malignancy.
Aminoglutethimide An adrenocortical steroid synthesis inhibitor used in the treatment of Cushing's syndrome.
Flutamide An antiandrogen used for locally confined stage B2-C and D-2 metastatic prostate carcinoma.
Toremifene A first generation nonsteroidal selective estrogen receptor modulator used to treat certain breast cancers.
Medroxyprogesterone acetate A progestin used as a contraceptive and in the treatment of secondary amenorrhea, abnormal uterine bleeding, pain from endometriosis, endometrial and renal carcinomas, paraphilia in males, and GnRH-dependent precocious puberty.
Prednisone A corticosteroid used to treat inflammation or immune-mediated reactions and to treat endocrine or neoplastic diseases.
Mitotane An adrenal cortex inhibitor used to treat adrenocortical tumors and Cushing's syndrome.
Tamoxifen A selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
Prednisolone A glucocorticoid used to treat adrenocortical insufficiency, inflammatory conditions, and some cancers.
Testolactone A medication used to treat advanced breast cancer.
Fulvestrant An estrogen receptor antagonist used to treat HR+ breast cancer that may also be HER2-.
Anastrozole A competitive, selective, non-steroidal aromatase inhibitor used as adjuvant therapy for the treatment of hormone receptor-positive breast cancer in postmenopausal women.
Dexamethasone A glucocorticoid available in various modes of administration that is used for the treatment of various inflammatory conditions, including bronchial asthma, as well as endocrine and rheumatic disorders.
Methyltestosterone A synthetic anabolic steroid used for the replacement therapy in conditions associated with testosterone deficiencies in males, such as hypogonadism, and treatment of advancing inoperable metastatic breast cancer in females.
Triptorelin A GnRH agonist indicated for the palliative treatment of advanced prostate cancer.
Hexestrol A synthetic estrogen that has been used as a hormonal antineoplastic agent.
Estramustine An antineoplastic agent used for the management of metastatic and/or progressive prostate cancer in palliative setting.
Tibolone For the relief of post-menopausal symptoms and for the prevention of osteoporosis .
Dienogest An oral progestin used for the treatment of endometriosis as monotherapy or contraception in combination with ethinylestradiol.
Liarozole Liarozole has been used in trials studying the treatment of Ichthyosis, Lamellar.
Methylprednisolone hemisuccinate 水溶性用类固醇激素治疗切断e allergic reactions, dermatologic diseases, endocrine disorders, gastrointestinal diseases, hematological disorders, neoplastic diseases, nervous system conditions, ophthalmic diseases, renal diseases, respiratory diseases, and rheumatic disorders.
Prednisone acetate Not Annotated
Estramustine phosphate A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.
Fadrozole Not Annotated
Drugs & Drug Targets
Drug Target Type
Leuprolide Gonadotropin-releasing hormone receptor target
Goserelin Lutropin-choriogonadotropic hormone receptor target
Goserelin Gonadotropin-releasing hormone receptor target
Octreotide Myeloperoxidase enzyme
Octreotide 阶段chrome P450 3A4 enzyme
Octreotide Somatostatin receptor target
Octreotide Serum albumin carrier
Octreotide P-glycoprotein 1 transporter
Octreotide Canalicular multispecific organic anion transporter 1 transporter
Diethylstilbestrol Estrogen receptor alpha target
Diethylstilbestrol Estrogen-related receptor gamma target
Diethylstilbestrol Transthyretin carrier
Diethylstilbestrol Catechol O-methyltransferase enzyme
Diethylstilbestrol 阶段chrome P450 19A1 enzyme
Diethylstilbestrol ATP-binding cassette sub-family G member 2 transporter
Diethylstilbestrol P-glycoprotein 1 transporter
Diethylstilbestrol Estrogen receptor beta target
Diethylstilbestrol 阶段chrome P450 3A4 enzyme
Diethylstilbestrol 阶段chrome P450 2C8 enzyme
Diethylstilbestrol 阶段chrome P450 2C9 enzyme
Diethylstilbestrol 阶段chrome P450 2E1 enzyme
Diethylstilbestrol Steroid hormone receptor ERR1 target
Diethylstilbestrol Steroid hormone receptor ERR2 target
Diethylstilbestrol Nuclear receptor coactivator 2 target
Diethylstilbestrol Nuclear receptor subfamily 1 group I member 2 target
Diethylstilbestrol Androgen receptor target
Diethylstilbestrol Sex hormone-binding globulin target
Diethylstilbestrol Solute carrier organic anion transporter family member 1B1 transporter
Diethylstilbestrol Solute carrier organic anion transporter family member 2B1 transporter
Diethylstilbestrol Bile salt export pump transporter
Chlorotrianisene Estrogen receptor alpha target
Chlorotrianisene 阶段chrome P450 19A1 enzyme
Megestrol acetate Progesterone receptor target
Megestrol acetate Glucocorticoid receptor target
Megestrol acetate P-glycoprotein 1 transporter
Megestrol acetate 阶段chrome P450 3A4 enzyme
Aminoglutethimide 阶段chrome P450 19A1 target
Aminoglutethimide 阶段chrome P450 2C19 enzyme
Aminoglutethimide 阶段chrome P450 3A4 enzyme
Aminoglutethimide Cholesterol side-chain cleavage enzyme, mitochondrial target
Flutamide Androgen receptor target
Flutamide 阶段chrome P450 1A2 enzyme
Flutamide 阶段chrome P450 3A4 enzyme
Flutamide 阶段chrome P450 1A1 enzyme
Flutamide 阶段chrome P450 1B1 enzyme
Flutamide 阶段chrome P450 3A5 enzyme
Flutamide Aryl hydrocarbon receptor target
Flutamide Nuclear receptor subfamily 1 group I member 2 target
Flutamide Multidrug resistance-associated protein 1 transporter
Toremifene Estrogen receptor alpha target
Toremifene 阶段chrome P450 3A4 enzyme
Toremifene P-glycoprotein 1 transporter
Toremifene 阶段chrome P450 1A1 enzyme
Toremifene Sex hormone-binding globulin target
Medroxyprogesterone acetate Progesterone receptor target
Medroxyprogesterone acetate Estrogen receptor alpha target
Medroxyprogesterone acetate 阶段chrome P450 3A4 enzyme
Medroxyprogesterone acetate 阶段chrome P450 2C8 enzyme
Medroxyprogesterone acetate 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2 enzyme
Medroxyprogesterone acetate 阶段chrome P450 2C9 enzyme
Medroxyprogesterone acetate 阶段chrome P450 3A1 enzyme
Medroxyprogesterone acetate Serum albumin carrier
Medroxyprogesterone acetate P-glycoprotein 1 target
Medroxyprogesterone acetate GABA(A) Receptor target
Medroxyprogesterone acetate P-glycoprotein 1 transporter
Prednisone Glucocorticoid receptor target
Prednisone 阶段chrome P450 3A4 enzyme
Prednisone P-glycoprotein 1 transporter
Prednisone Solute carrier organic anion transporter family member 1A2 transporter
Prednisone 阶段chrome P450 2C19 enzyme
Prednisone Serum albumin carrier
Prednisone 阶段chrome P450 3A5 enzyme
Prednisone Corticosteroid-binding globulin carrier
Prednisone 阶段chrome P450 3A Subfamily enzyme
Prednisone 阶段chrome P450 2A6 enzyme
Prednisone 阶段chrome P450 1B1 enzyme
Prednisone 阶段chrome P450 2B6 enzyme
Prednisone 阶段chrome P450 2C8 enzyme
Prednisone 阶段chrome P450 2C9 enzyme
Prednisone Corticosteroid 11-beta-dehydrogenase isozyme 1 enzyme
Mitotane 阶段chrome P450 11B1, mitochondrial target
Mitotane Adrenodoxin, mitochondrial target
Mitotane Sex hormone-binding globulin carrier
Mitotane Corticosteroid-binding globulin carrier
Mitotane 阶段chrome P450 3A4 enzyme
Mitotane Estrogen receptor alpha target
Mitotane Progesterone receptor target
Mitotane Androgen receptor target
Mitotane Thyroxine-binding globulin carrier
Mitotane P-glycoprotein 1 transporter
Tamoxifen Estrogen receptor alpha target
Tamoxifen Estrogen receptor beta target
Tamoxifen 阶段chrome P450 2C9 enzyme
Tamoxifen 阶段chrome P450 3A4 enzyme
Tamoxifen 阶段chrome P450 2D6 enzyme
Tamoxifen 阶段chrome P450 2C8 enzyme
Tamoxifen 阶段chrome P450 2B6 enzyme
Tamoxifen Liver carboxylesterase 1 enzyme
Tamoxifen 阶段chrome P450 3A5 enzyme
Tamoxifen 阶段chrome P450 1A1 enzyme
Tamoxifen 阶段chrome P450 1B1 enzyme
Tamoxifen 阶段chrome P450 2C19 enzyme
Tamoxifen Dimethylaniline monooxygenase [N-oxide-forming] 1 enzyme
Tamoxifen Dimethylaniline monooxygenase [N-oxide-forming] 3 enzyme
Tamoxifen 阶段chrome P450 3A7 enzyme
Tamoxifen P-glycoprotein 1 transporter
Tamoxifen ATP-binding cassette sub-family G member 2 transporter
Tamoxifen 阶段chrome P450 19A1 enzyme
Tamoxifen 阶段chrome P450 2A6 enzyme
Tamoxifen 阶段chrome P450 2E1 enzyme
Tamoxifen UDP-glucuronosyltransferase 1-10 enzyme
Tamoxifen Sulfotransferase 1A1 enzyme
Tamoxifen Canalicular multispecific organic anion transporter 1 transporter
Tamoxifen 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase target
Tamoxifen Protein kinase C target
Tamoxifen Androgen receptor target
Tamoxifen Potassium voltage-gated channel subfamily H member 2 target
Tamoxifen Nuclear receptor subfamily 1 group I member 2 target
Tamoxifen Estrogen-related receptor gamma target
Tamoxifen Sex hormone-binding globulin target
Tamoxifen Bile salt export pump transporter
Tamoxifen Thyroxine-binding globulin carrier
Tamoxifen Bile salt sulfotransferase enzyme
Tamoxifen 阶段chrome P450 1A2 enzyme
Tamoxifen UDP-glucuronosyltransferase 2B7 enzyme
Tamoxifen UDP-glucuronosyltransferase 2B17 enzyme
Tamoxifen Estrogen sulfotransferase enzyme
Tamoxifen ATP-binding cassette sub-family A member 1 transporter
Tamoxifen Mitogen-activated protein kinase 8 target
Tamoxifen Serum albumin carrier
Prednisolone Corticosteroid-binding globulin carrier
Prednisolone 阶段chrome P450 3A4 enzyme
Prednisolone Glucocorticoid receptor target
Prednisolone Solute carrier organic anion transporter family member 1A2 transporter
Prednisolone P-glycoprotein 1 transporter
Prednisolone Serum albumin carrier
Testolactone 阶段chrome P450 19A1 target
Fulvestrant Estrogen receptor alpha target
Fulvestrant 阶段chrome P450 3A4 enzyme
Fulvestrant UDP-glucuronosyltransferase 1-1 enzyme
Anastrozole 阶段chrome P450 19A1 target
Anastrozole P-glycoprotein 1 transporter
Anastrozole 阶段chrome P450 3A4 enzyme
Anastrozole 阶段chrome P450 3A5 enzyme
Anastrozole 阶段chrome P450 2C8 enzyme
Anastrozole UDP-glucuronosyltransferase 1-4 enzyme
Anastrozole UDP-glucuronosyltransferase 1-3 enzyme
Anastrozole UDP-glucuronosyltransferase 2B7 enzyme
Anastrozole 阶段chrome P450 1A2 enzyme
Anastrozole 阶段chrome P450 2C9 enzyme
Dexamethasone Glucocorticoid receptor target
Dexamethasone Annexin A1 target
Dexamethasone Nitric oxide synthase, inducible target
Dexamethasone Nuclear receptor subfamily 0 group B member 1 target
Dexamethasone 阶段chrome P450 3A4 enzyme
Dexamethasone 阶段chrome P450 3A5 enzyme
Dexamethasone 阶段chrome P450 3A7 enzyme
Dexamethasone Bile salt export pump transporter
Dexamethasone P-glycoprotein 1 transporter
Dexamethasone Canalicular multispecific organic anion transporter 1 transporter
Dexamethasone Solute carrier organic anion transporter family member 1A2 transporter
Dexamethasone ATP-binding cassette sub-family G member 2 transporter
Dexamethasone Steroid 17-alpha-hydroxylase/17,20 lyase enzyme
Dexamethasone 阶段chrome P450 1A1 enzyme
Dexamethasone 阶段chrome P450 2A6 enzyme
Dexamethasone 阶段chrome P450 2B6 enzyme
Dexamethasone 阶段chrome P450 2C19 enzyme
Dexamethasone 阶段chrome P450 2C8 enzyme
Dexamethasone 阶段chrome P450 2E1 enzyme
Dexamethasone 阶段chrome P450 3A43 enzyme
Dexamethasone 阶段chrome P450 4A11 enzyme
Dexamethasone Nuclear receptor subfamily 1 group I member 2 target
Dexamethasone 阶段chrome P450 11B1, mitochondrial enzyme
Dexamethasone Serum albumin carrier
Dexamethasone Corticosteroid 11-beta-dehydrogenase isozyme 2 enzyme
Dexamethasone Corticosteroid 11-beta-dehydrogenase isozyme 1 enzyme
Dexamethasone Solute carrier family 22 member 8 transporter
Methyltestosterone 阶段chrome P450 2B6 enzyme
Methyltestosterone 阶段chrome P450 3A4 enzyme
Methyltestosterone Androgen receptor target
Methyltestosterone Solute carrier organic anion transporter family member 1A2 transporter
Methyltestosterone Solute carrier family 22 member 8 transporter
Methyltestosterone Serum albumin carrier
Methyltestosterone Sex hormone-binding globulin carrier
Methyltestosterone Estrogen receptor alpha target
Methyltestosterone 阶段chrome P450 19A1 enzyme
Triptorelin Gonadotropin-releasing hormone receptor target
Hexestrol Aldo-keto reductase family 1 member C1 target
Hexestrol Estrogen receptor alpha target
Hexestrol Nuclear receptor subfamily 1 group I member 2 target
Hexestrol Nuclear receptor subfamily 1 group I member 3 target
Estramustine Estrogen receptor beta target
Estramustine Estrogen receptor alpha target
Estramustine Microtubule-associated protein 2 target
Estramustine Microtubule-associated蛋白1 target
Estramustine P-glycoprotein 1 transporter
Estramustine 阶段chrome P450 3A4 enzyme
Tibolone Estrogen receptor alpha target
Tibolone Steryl-sulfatase enzyme
Tibolone 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 enzyme
Tibolone 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2 enzyme
Tibolone Sulfotransferase 1A1 enzyme
Tibolone Serum albumin carrier
Dienogest 阶段chrome P450 3A4 enzyme
Dienogest Progesterone receptor target
Dienogest Androgen receptor target
Methylprednisolone hemisuccinate 阶段chrome P450 3A4 enzyme
Methylprednisolone hemisuccinate 阶段chrome P450 3A5 enzyme
Prednisone acetate 阶段chrome P450 3A4 enzyme
Prednisone acetate 阶段chrome P450 3A5 enzyme