Selective Immunosuppressants

Name
Selective Immunosuppressants
Accession Number
DBCAT002129
Description

Not Available

ATC Classification
Drugs
Drug Drug Description
Muromonab A monoclonal anti-CD3 antibody used as immunosuppressive therapy in kidney, heart, and liver transplant patients.
Alemtuzumab A monoclonal anti-CD52 antibody used in the treatment of B-cell chronic lymphocytic leukemia and relapsing forms of multiple sclerosis.
Alefacept A recombinant fusion protein that binds CD2 and is used treat moderate to severe plaque psoriasis.
Efalizumab A monoclonal anti-CD11a antibody used to treat moderate to severe plaque psoriasis.
Antithymocyte immunoglobulin (rabbit) A purified form of rabbit anti-thymocyte antibodies used for immunosuppression in patients receiving kidney transplants.
Natalizumab A monoclonal anti-integrin antibody which binds to the alpha 4 subunit of integrins to prevent migration of immune cells, and is used to treat Crohn's disease or multiple sclerosis.
Sirolimus An mTOR inhibitor immunosuppressant used to prevent organ transplant rejections, treat lymphangioleiomyomatosis, and treat adults with perivascular epithelioid cell tumors.
Mycophenolic acid An immunosuppressant used to prevent organ transplant rejections.
Leflunomide A pyrimidine synthesis inhibitor indicated to treat rheumatoid arthritis.
Eculizumab A recombinant humanized monoclonal antibody used to reduce the risk of hemolysis in paroxysmal nocturnal hemoglobinuria (PNH) and atypical hemolytic uremic syndrome (aHUS).
Abatacept A disease-modifying antirheumatic drug (DMARD) used in the management of rheumatic conditions, such as rheumatoid or psoriatic arthritis, and for the prophylaxis of acute graft-versus-host disease.
Everolimus A mammalian target of rapamycin (mTOR) kinase inhibitor used to treat various types of malignancies.
Apremilast 非甾体类药物用于治疗of inflammatory conditions such as psoriasis and psoriatic arthritis.
Abetimus 追究在kidn使用/治疗ey disease and systemic lupus erythematosus.
Belatacept A selective T-cell costimulation blocker used in the prophylaxis of organ rejection in adult patients receiving a kidney transplant.
Fingolimod A sphingosine 1-phosphate receptor modulator used to treat patients with the relapsing-remitting form of multiple sclerosis (MS) and studied to manage lung complications of COVID-19.
Belimumab A B-lymphocyte stimulator (BLyS)-specific inhibitor that indirectly inhibits B cell survival, and is used to treat patients with autoantibody positive, active systemic lupus erythematosus.
Teriflunomide A pyrimidine synthesis inhibitor with anti-inflammatory and immunomodulatory properties used to treat patients with the relapsing-remitting form of multiple sclerosis.
Tofacitinib A Janus kinase (JAK) inhibitor used to treat rheumatic conditions, such as rheumatoid arthritis and ankylosing spondylitis, and ulcerative colitis.
Vedolizumab An integrin blocker and anti-inflammatory agent used to manage ulcerative colitis and Crohn's disease in adults with inadequate clinical response to immunomodulators.
Antilymphocyte immunoglobulin (horse) A primarily IgG immune globulin used to manage allograft rejection in renal transplant patients.
Gusperimus Gusperimus has been used in trials studying the treatment of Lupus Nephritis, Wegeners Granulomatosis, and Wegener's Granulomatosis.
Begelomab Not Annotated
Cladribine A purine antimetabolite used for the management of relapsing forms of Multiple Sclerosis (MS), used in patients who have not responded to or who were unable to tolerate alternative MS drugs.
Baricitinib A Janus kinase inhibitor used to treat moderate to severe rheumatoid arthritis that has responded poorly to at least one TNF antagonist.
Ocrelizumab A CD20 specific monoclonal antibody used to treat relapsing remitting multiple sclerosis.
Ozanimod A sphingosine 1-phosphate receptor modulator being studied to treat Multiple Sclerosis (MS) and inflammatory bowel disease (IBD).
Emapalumab An interferon gamma blocking antibody used to treat primary hemophagocytic lymphohistiocytosis.
Risankizumab An interleukin-23 antagonist used to treat moderate to severe plaque psoriasis, active psoriatic arthritis, and moderately to severely active Crohn's disease in adults.
Ravulizumab A monoclonal antibody used to treat paroxysmal nocturnal hemoglobinuria, atypical hemolytic uremic syndrome, and myasthenia gravis.
Siponimod A medication used to treat relapsing multiple sclerosis.
Upadacitinib An oral Janus kinase (JAK)1-selective inhibitor used in the treatment of moderate to severe rheumatoid arthritis, active psoriatic arthritis, ankylosing spondylitis, and severe atopic dermatitis, including in patients who did not respond well to other therapies.
Imlifidase A cysteine protease that specifically cleaves human IgG antibodies, facilitating kidney transplantation in HLA sensitized patients.
Drugs & Drug Targets
Drug Target Type
Muromonab T-cell surface glycoprotein CD3 epsilon chain target
Muromonab Low affinity immunoglobulin gamma Fc region receptor III-B target
Muromonab T-cell surface glycoprotein CD3 delta chain target
Muromonab T-cell surface glycoprotein CD3 gamma chain target
Muromonab T-cell surface glycoprotein CD3 zeta chain target
Alemtuzumab CAMPATH-1 antigen target
Alemtuzumab Low affinity immunoglobulin gamma Fc region receptor III-B target
Alemtuzumab Low affinity immunoglobulin gamma Fc region receptor III-A target
Alemtuzumab High affinity immunoglobulin gamma Fc receptor I target
Alemtuzumab Low affinity immunoglobulin gamma Fc region receptor II-a target
Alemtuzumab Low affinity immunoglobulin gamma Fc region receptor II-b target
Alemtuzumab Low affinity immunoglobulin gamma Fc region receptor II-c target
Alefacept T-cell surface antigen CD2 target
Alefacept Low affinity immunoglobulin gamma Fc region receptor III-B target
Alefacept Low affinity immunoglobulin gamma Fc region receptor III-A target
Efalizumab Integrin alpha-L target
Efalizumab Integrin alpha-X target
Antithymocyte immunoglobulin (rabbit) T-cell surface glycoprotein CD1a target
Antithymocyte immunoglobulin (rabbit) Major histocompatibility complex class I-related gene protein target
Antithymocyte immunoglobulin (rabbit) Integrin alpha-L target
Antithymocyte immunoglobulin (rabbit) T-lymphocyte activation antigen CD86 target
Antithymocyte immunoglobulin (rabbit) Low affinity immunoglobulin gamma Fc region receptor II-b target
Antithymocyte immunoglobulin (rabbit) T-cell surface glycoprotein CD4 target
Antithymocyte immunoglobulin (rabbit) Integrin beta-1 target
Antithymocyte immunoglobulin (rabbit) Integrin alpha-V target
Antithymocyte immunoglobulin (rabbit) Integrin beta-3 target
Natalizumab Integrin alpha-4 target
Natalizumab Low affinity immunoglobulin gamma Fc region receptor III-B target
Natalizumab High affinity immunoglobulin gamma Fc receptor I target
Natalizumab Intercellular adhesion molecule 1 target
Sirolimus Cytochrome P450 3A4 enzyme
Sirolimus Serine/threonine-protein kinase mTOR target
Sirolimus Cytochrome P450 3A5 enzyme
Sirolimus Cytochrome P450 3A7 enzyme
Sirolimus P-glycoprotein 1 transporter
Sirolimus Solute carrier organic anion transporter family member 1B1 transporter
Sirolimus Multidrug and toxin extrusion protein 1 transporter
Sirolimus Serum albumin carrier
Sirolimus Alpha-1-acid glycoprotein 1 carrier
Sirolimus Apolipoproteins carrier
Mycophenolic acid Inosine-5'-monophosphate dehydrogenase 2 target
Mycophenolic acid Inosine-5'-monophosphate dehydrogenase 1 target
Mycophenolic acid UDP-glucuronosyltransferase 1-1 enzyme
Mycophenolic acid UDP-glucuronosyltransferase 1-9 enzyme
Mycophenolic acid UDP-glucuronosyltransferase 2B7 enzyme
Mycophenolic acid UDP-glucuronosyltransferase 1-7 enzyme
Mycophenolic acid UDP-glucuronosyltransferase 1-6 enzyme
Mycophenolic acid Serum albumin carrier
Mycophenolic acid UDP-glucuronosyltransferase 1-8 enzyme
Mycophenolic acid UDP-glucuronosyltransferase 1-10 enzyme
Mycophenolic acid Cytochrome P450 3A4 enzyme
Mycophenolic acid Cytochrome P450 3A5 enzyme
Mycophenolic acid Cytochrome P450 2C8 enzyme
Leflunomide Dihydroorotate dehydrogenase (quinone), mitochondrial target
Leflunomide Cytochrome P450 1A2 enzyme
Leflunomide Cytochrome P450 2C9 enzyme
Leflunomide Aryl hydrocarbon receptor target
Leflunomide Protein-tyrosine kinase 2-beta target
Leflunomide ATP-binding cassette sub-family G member 2 transporter
Eculizumab Complement C5 target
Abatacept T-lymphocyte activation antigen CD80 target
Abatacept T-lymphocyte activation antigen CD86 target
Abatacept Cytotoxic T-lymphocyte protein 4 target
Everolimus Serine/threonine-protein kinase mTOR target
Everolimus Cytochrome P450 3A4 enzyme
Everolimus Solute carrier organic anion transporter family member 1B1 transporter
Everolimus Solute carrier organic anion transporter family member 1B3 transporter
Everolimus Solute carrier organic anion transporter family member 1A2 transporter
Everolimus Cytochrome P450 2D6 enzyme
Everolimus P-glycoprotein 1 transporter
Apremilast Phosphodiesterase isozyme 4 target
Apremilast Cytochrome P450 3A4 enzyme
Apremilast Cytochrome P450 2A6 enzyme
Apremilast Cytochrome P450 1A2 enzyme
Apremilast P-glycoprotein 1 transporter
Belatacept T-lymphocyte activation antigen CD86 target
Belatacept T-lymphocyte activation antigen CD80 target
Fingolimod Sphingosine 1-phosphate receptor 5 target
Fingolimod Sphingosine kinase 1 enzyme
Fingolimod Cytochrome P450 2E1 enzyme
Fingolimod Leukotriene-B(4) omega-hydroxylase 1 enzyme
Fingolimod Histone deacetylase 1 target
Fingolimod Excitatory amino acid transporter 2 transporter
Fingolimod Excitatory amino acid transporter 1 transporter
Fingolimod P-glycoprotein 1 transporter
Fingolimod 耐多药resistance-associated蛋白质1 transporter
Fingolimod Sphingosine 1-phosphate receptor 1 target
Fingolimod Sphingosine 1-phosphate receptor 4 target
Fingolimod Sphingosine 1-phosphate receptor 3 target
Belimumab Tumor necrosis factor ligand superfamily member 13B target
Teriflunomide ATP-binding cassette sub-family G member 2 transporter
Teriflunomide Dihydroorotate dehydrogenase (quinone), mitochondrial target
Teriflunomide Cytochrome P450 2C8 enzyme
Teriflunomide Solute carrier organic anion transporter family member 1B1 transporter
Teriflunomide Cytochrome P450 1A2 enzyme
Tofacitinib Non-receptor tyrosine-protein kinase TYK2 target
Tofacitinib Cytochrome P450 3A4 enzyme
Tofacitinib Cytochrome P450 2C19 enzyme
Tofacitinib Tyrosine-protein kinase JAK2 target
Tofacitinib Tyrosine-protein kinase JAK1 target
Tofacitinib Tyrosine-protein kinase JAK3 target
Tofacitinib Serum albumin carrier
Vedolizumab Integrin alpha-4 target
Vedolizumab Integrin beta-7 target
Cladribine Purine nucleoside phosphorylase target
Cladribine DNA target
Cladribine Deoxycytidine kinase enzyme
Cladribine Ribonucleoside-diphosphate reductase large subunit target
Cladribine Ribonucleoside-diphosphate reductase subunit M2 target
Cladribine Ribonucleoside-diphosphate reductase subunit M2 B target
Cladribine DNA polymerase alpha catalytic subunit target
Cladribine DNA polymerase epsilon catalytic subunit A target
Cladribine DNA polymerase epsilon subunit 2 target
Cladribine DNA polymerase epsilon subunit 3 target
Cladribine DNA polymerase epsilon subunit 4 target
Cladribine ATP-binding cassette sub-family G member 2 transporter
Cladribine Solute carrier family 28 member 3 transporter
Baricitinib Solute carrier family 22 member 8 transporter
Baricitinib ATP-binding cassette sub-family G member 2 transporter
Baricitinib Multidrug and toxin extrusion protein 2 transporter
Baricitinib Cytochrome P450 3A4 enzyme
Baricitinib Tyrosine-protein kinase JAK1 target
Baricitinib Tyrosine-protein kinase JAK2 target
Baricitinib Solute carrier family 22 member 6 transporter
Baricitinib Solute carrier family 22 member 2 transporter
Baricitinib Solute carrier organic anion transporter family member 1B3 transporter
Baricitinib Tyrosine-protein kinase JAK3 target
Baricitinib P-glycoprotein 1 transporter
Baricitinib Non-receptor tyrosine-protein kinase TYK2 target
Ocrelizumab B-lymphocyte antigen CD20 target
Ozanimod Sphingosine 1-phosphate receptor 1 target
Ozanimod Sphingosine 1-phosphate receptor 5 target
Ozanimod Amine oxidase [flavin-containing] B transporter
Ozanimod ATP-binding cassette sub-family G member 2 transporter
Ozanimod P-glycoprotein 1 transporter
Ozanimod Fatty aldehyde dehydrogenase enzyme
Ozanimod Alcohol dehydrogenase class-3 enzyme
Ozanimod Arylamine N-acetyltransferase 2 enzyme
Ozanimod Cytochrome P450 2C8 enzyme
Ozanimod Amine oxidase [flavin-containing] B enzyme
Ozanimod Aldo-keto reductase family 1 member C1 enzyme
Ozanimod Aldo-keto reductase family 1 member C2 enzyme
Ozanimod Cytochrome P450 3A4 enzyme
Emapalumab Interferon gamma target
Risankizumab Interleukin-23 target
Ravulizumab Complement C5 target
Siponimod Sphingosine 1-phosphate receptor 5 target
Siponimod Sphingosine 1-phosphate receptor 1 target
Siponimod Cytochrome P450 3A4 enzyme
Siponimod Cytochrome P450 2C9 enzyme
Upadacitinib Tyrosine-protein kinase JAK1 target
Upadacitinib Cytochrome P450 3A4 enzyme
Upadacitinib Cytochrome P450 2D6 enzyme
Upadacitinib P-glycoprotein 1 transporter
Upadacitinib ATP-binding cassette sub-family G member 2 transporter
Upadacitinib Solute carrier organic anion transporter family member 1B1 transporter
Imlifidase IgG heavy chain target